Signal Transduction and Targeted Therapy: PAK1 is a broad-spectrum anti-SARS-CoV-2 target

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2), the causative agent of coronavirus disease 2019 (COVID-19), has had a significant impact on healthcare systems and economies worldwide. The emergence of new viral strains represents a major challenge in the development of effective antiviral agents. The spike protein of SARS-CoV-2 interacts with ACE2 on the cell surface, facilitating viral attachment and entry. Spike protein also promotes ACE2 degradation, but the molecular mechanisms are not fully determined. In this study, Dr. Ming Liu et al from our laboratory showed that the spike-ACE2 complex is endocytosed and degraded via autophagy, in a manner that depends on clathrin-mediated endocytosis and PAK1-mediated cytoskeleton rearrangement. Importantly, through collaboration with ...read more